product summary
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company name :
Tocris Bioscience
product type :
chemical
product name :
SJPYT 310
catalog :
8839/10
quantity :
10 mg (also 50 mg)
price :
143 USD
more info or order :
Tocris Bioscience product webpage
product information
brand :
Tocris
catalog number base :
8839
SKU :
8839/10
product name :
SJPYT 310
units size :
10 mg (also 50 mg)
description :
Potent and selective PXR antagonist
target :
PXR/NR1I2
category :
Small Molecules
purity :
98%
observed molecular weight :
464.61
url print :
?utm_source=biocompare&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules
details of functionality :
SJPYT 310 is a potent and selective PXR antagonist (IC50 values are 4 and 9 nM for binding and cellular activity, respectively). SJPYT 310 displays selectivity for hPXR without affecting the activity of mPXR, hCAR, hFXR, hLXR , or hVDR. SJPYT 310 shows no toxicity.
top caption :
Potent and selective PXR antagonist
extended description :
Potent and selective PXR antagonist
chemical name text :
N-[5-(1,1-Dimethylethyl)-2-[(1S)-1-methylbutoxy]phenyl]-1-(2-methoxy-5-methylphenyl)-5-methyl-1H-1,2,3-triazole-4-carboxamide
formula :
C27H36N4O3
formula text :
C27H36N4O3
cas num :
2883814-84-2
USD :
143 USD
product details :
Potent and selective PXR antagonist
alt names :
BXR, NR1I2, nuclear receptor subfamily 1 group I member 2, nuclear receptor subfamily 1, group I, member 2, ONR1, Orphan nuclear receptor PAR1, Orphan nuclear receptor PXR, PAR, PAR1, PAR2, Pregnane X receptor, PRR, PXRPARq, SAR, Steroid and xenobiotic receptor, SXR, SXRBXR
storage :
Store at -20°C
more info or order :
Tocris Bioscience product webpage
company information
Tocris Bioscience
The Watkins Building
Atlantic Road
Avonmouth, Bristol
BS11 9QD
info@bio-techne.com
https://www.tocris.com
800-343-7475
headquarters: UK