8095/1 | Tocris Bioscience 8095/1 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

8095/1

catalog :

8095/1

quantity :

1 mg

price :

140 USD

more info or order :

Tocris Bioscience product webpage

image

image 1 :

Atypical chemokine receptor (ACKR3) agonist

product information

master code :

8095

SKU :

8095/1

product name :

LIH 383

unit size :

1 mg

description :

Atypical chemokine receptor (ACKR3) agonist

target :

Chemokine Receptor Agonists

category :

Peptides

purity :

95%

observed molecular weight :

997.23

url print :

?utm_source=labome&utm_medium=referral&utm_campaign=product&utm_term=peptides

details of functionality :

LIH 383 is a potent and highly selective atypical chemokine receptor (ACKR3/CXCR7) agonist. LIH 383 competes directly with CXCL12-AF647 and is more potent in inducing -arrestin recruitment to ACKR3 (EC50 = 0.61 nM) than the full-length chemokine ligands CXCL12 or CXCL11 (EC50 values are 1.2 nM and 2.2 nM, respectively). In a rat ex vivo model, LIH 383 increases the availability and signaling of opioid peptides at classical receptors.

top caption :

Atypical chemokine receptor (ACKR3) agonist

extended description :

Atypical chemokine receptor (ACKR3) agonist

formula :

C45H72N16O8S

formula text :

C45H72N16O8S

cas num :

2866266-58-0

USD :

140 USD

product details :

Atypical chemokine receptor (ACKR3) agonist

storage :

Store at -20░C

more info or order :

Tocris Bioscience product webpage