8055/10 | Tocris Bioscience 8055/10 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

8055/10

catalog :

8055/10

quantity :

10 mg (also 50 mg)

price :

195 USD

more info or order :

Tocris Bioscience product webpage

image

image 1 :

M5 Muscarinic Acetylcholine Receptor Antagonist

product information

master code :

8055

SKU :

8055/10

product name :

VU 6019650

unit size :

10 mg (also 50 mg)

description :

M5 receptor antagonist

target :

mAChR M5 Antagonists

category :

Small Molecules

purity :

98%

observed molecular weight :

411.51

url print :

?utm_source=labome&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

VU 6019650 is a potent and selective M5 receptor antagonist (hM5 IC50 = 36 nM). Exhibits 100-fold selectivity over human and rat M1-4. In vivo , VU 6019650 inhibits the reward effects of oxycodone and reduces oxycodone self-administration in rats. VU 6019650 is blood brain barrier penetrant.

top caption :

M5 Muscarinic Acetylcholine Receptor Antagonist

extended description :

M5 receptor antagonist

chemical name text :

(3R,4S)-rel-1-[(2,3-Dihydro-5-benzofuranyl)sulfonyl]-3-fluoro-4-[[(1-methyl-1H-imidazol-2-yl)thio]methyl]piperidine

formula :

C18H22FN3O3S2

formula text :

C18H22FN3O3S2

cas num :

2926782-31-0

USD :

195 USD

product details :

M5 receptor antagonist

alt names :

cholinergic receptor, muscarinic 5, HM5, M5, M5R, mAChR M5, MGC41838, muscarinic acetylcholine receptor M5

storage :

Store at -20░C

more info or order :

Tocris Bioscience product webpage