7927/10 | Tocris Bioscience 7927/10 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

7927/10

catalog :

7927/10

quantity :

10 mg (also 50 mg)

price :

199 USD

more info or order :

Tocris Bioscience product webpage

image

image 1 :

Potent and selective SRPK family inhibitor

product information

master code :

7927

SKU :

7927/10

product name :

MSC 1186

unit size :

10 mg (also 50 mg)

description :

Potent and selective SRPK family inhibitor

target :

SRPK3

category :

Small Molecules

purity :

98%

observed molecular weight :

461.9

url print :

?utm_source=labome&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

MSC1186 is a potent and selective inhibitor of serine arginine protein kinases (SRPK) 3, 1 and 2 (IC50 values are 0.6 nM, 3 nM and 81 nM respectively in biochemical assay; EC50 values in NanoBRETassay are 40 nM, 98 nM and 149 nM, respectively). Shows no activity at CLK and DYRK families (IC50 10 M).

top caption :

Potent and selective SRPK family inhibitor

extended description :

Potent and selective SRPK family inhibitor

chemical name text :

N-[3-[[[2-(6-Chloro-7-fluoro-1H-benzimidazol-2-yl)-4-pyrimidinyl]amino]methyl]-2-pyridinyl]-N-methylmethanesulfonamide

formula :

C19H17ClFN7O2S

formula text :

C19H17ClFN7O2S

cas num :

2871698-23-4

USD :

199 USD

product details :

Potent and selective SRPK family inhibitor

alt names :

MGC102944, MSSK1, MSSK-1, MSSK1EC 2.7.11.1, Muscle-specific serine kinase 1, serine arginine rich protein-specific kinase 3, Serine/arginine-rich protein-specific kinase 3, serine/threonine kinase 23, Serine/threonine-protein kinase 23, serine/threonine-protein kinase SRPK3, SFRS protein kinase 3, SFRSK2, SR-protein-specific kinase 3, SRSF protein kinase 3, STK23

storage :

Store at -20░C

more info or order :

Tocris Bioscience product webpage