7926/250 | Tocris Bioscience 7926/250 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

7926/250

catalog :

7926/250

quantity :

250 mg

price :

63 USD

more info or order :

Tocris Bioscience product webpage

image

image 1 :

Selective orthostatic agonist of hFFA2-DREADDs

product information

master code :

7926

SKU :

7926/250

product name :

MOMBA

unit size :

250 mg

description :

Selective orthostatic agonist of hFFA2-DREADDs

target :

DREADD Activators

category :

Small Molecules

purity :

98%

observed molecular weight :

166.17

url print :

?utm_source=labome&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

MOMBA is a selective orthosteric agonist for human free fatty acid 2 (hFFA2) engineered receptors, designer receptors activated by designer drugs (DREADD), it shows no activity to wild-type hFFA2, hFFA3, and mouse FFA2. MOMBA inhibit forskolin-stimulated cAMP levels in cells expressing the hFFA2-DREADD receptor with improved potency and equivalent efficacy to Sorbic acid (Cat. No. 7119). In hFFA2-DREADD transgenic mice, MOMBA treatment significantly reduces gut transit and promotes concentration-dependent release of GLP-1 from colonic crypts. Orally bioavailable.

top caption :

Selective orthostatic agonist of hFFA2-DREADDs

extended description :

Selective orthostatic agonist of hFFA2-DREADDs

chemical name text :

4-Methoxy-3-methylbenzoic acid

formula :

C9H10O3

formula text :

C9H10O3

cas num :

4/2/80

USD :

63 USD

product details :

Selective orthostatic agonist of hFFA2-DREADDs

storage :

Store at -20░C

more info or order :

Tocris Bioscience product webpage