7879/5 | Tocris Bioscience 7879/5 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

7879/5

catalog :

7879/5

quantity :

5 mg

price :

187 USD

more info or order :

Tocris Bioscience product webpage

image

image 1 :

Potent and selective HDAC class IIa inhibitor

product information

master code :

7879

SKU :

7879/5

product name :

CHDI 00484077

unit size :

5 mg

description :

Potent and selective HDAC class IIa inhibitor

target :

Class II Histone Deacetylases Inhibitors

category :

Small Molecules

purity :

98%

observed molecular weight :

382.39

url print :

?utm_source=labome&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

CHDI 00484077 is a potent and selective class IIa histone deacetylase HDAC inhibitor (IC50 values = 10-30 nM in vivo , 0.01 nM and 0.04 nM in HEK293 and Jurkat cells, respectively). Exhibits 150-fold selectivity for class IIa over class I/IIb HDACs in cells. Orally bioavailable and CNS penetrant.

top caption :

Potent and selective HDAC class IIa inhibitor

extended description :

Potent and selective HDAC class IIa inhibitor

chemical name text :

N-((R)-1-((S)-2-Methylpyrrolidin-1-yl)propan-2-yl)-4-(5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl)benzamide

formula :

C18H21F3N4O2

formula text :

C18H21F3N4O2

cas num :

3025894-92-9

USD :

187 USD

product details :

Potent and selective HDAC class IIa inhibitor

storage :

Store at -20░C

more info or order :

Tocris Bioscience product webpage