7800/2 | Tocris Bioscience 7800/2 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

7800/2

catalog :

7800/2

quantity :

2 mg

price :

369 USD

more info or order :

Tocris Bioscience product webpage

image

image 1 :

Potent and selective CDK2 degrader (PROTAC )

product information

master code :

7800

SKU :

7800/2

product name :

CPS2

unit size :

2 mg

description :

Potent and selective CDK2 Degrader (PROTAC )

target :

Active Degraders

category :

Small Molecules

purity :

98%

observed molecular weight :

890.95

url print :

?utm_source=labome&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

CPS2 is a potent and selective CDK2 Degrader (PROTAC ) (IC50 = 24 nM). It induces CDK2 degradation in several AML cell lines, including NB4, U937, OCI-AML2, OCI-AML3 and Kasumi-1 cells. It induces differentiation of AML cell lines, primary AML cells, and granulocytic differentiation of HSCs. . PROTAC is a registered trademark of Arvinas Operations, Inc., and is used under license .

top caption :

Potent and selective CDK2 degrader (PROTAC )

extended description :

Potent and selective CDK2 Degrader (PROTAC )

chemical name text :

4-[[5-Amino-1-[(3-methyl-2-thienyl)carbonyl]-1H-1,2,4-triazol-3-yl]amino]-N-[2-[[1-[2-[2-[2-[[2-(2,6-dioxo-3-piperidinyl)-2,3-dihydro-1,3-dioxo-1H-isoindol-4-yl]amino]ethoxy]ethoxy]ethyl]-1H-1,2,3-triazol-4-yl]methoxy]ethyl]benzenesulfonamide

formula :

C38H42N12O10S2

formula text :

C38H42N12O10S2

cas num :

2756741-90-7

USD :

369 USD

product details :

Potent and selective CDK2 Degrader (PROTAC )

storage :

Store at -20░C

more info or order :

Tocris Bioscience product webpage