7667/50 | Tocris Bioscience 7667/50 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

7667/50

catalog :

7667/50

quantity :

50 mg

price :

121 USD

more info or order :

Tocris Bioscience product webpage

image

image 1 :

Cat.No. 7667 - Pimavanserin C25H34FN3O2 CAS No. 706779-91-1

product information

master code :

7667

SKU :

7667/50

product name :

Pimavanserin

unit size :

50 mg

description :

Selective 5-HT2A inverse agonist

target :

5-HT2A Receptor Antagonists

category :

Small Molecules

purity :

98%

observed molecular weight :

427.56

url print :

?utm_source=labome&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Pimavanserin (also known as ACP-103) is a selective, potent 5-HT2A receptor inverse agonist (IC50 = 2 nM). Pimavanserin displays ~ 40-fold higher affinity for 5-HT2A over 5-HT2C receptor. Chronic administration of Pimavanserin, suppresses amyloid- production and improves anxiety-related behavior and memory in Alzheimer s disease mouse models. Pimavanserin shows protective effects on midbrain dopaminergic neurons in a rat model of Parkinson s Disease.

top caption :

Selective 5-HT2A inverse agonist

extended description :

Selective 5-HT2A inverse agonist

chemical name text :

N-[(4-Fluorophenyl)methyl]-N-(1-methyl-4-piperidinyl)-N -[[4-(2-methylpropoxy)phenyl]methyl]urea

formula :

C25H34FN3O2

formula text :

C25H34FN3O2

cas num :

706779-91-1

USD :

121 USD

product details :

Selective 5-HT2A inverse agonist

storage :

Store at -20░C

more info or order :

Tocris Bioscience product webpage