7658/10 | Tocris Bioscience 7658/10 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

7658/10

catalog :

7658/10

quantity :

10 mg (also 50 mg)

price :

281 USD

more info or order :

Tocris Bioscience product webpage

image

image 1 :

Cat.No. 7658 - VU 6028418 hydrochloride C23H27F3N4O.HCl

product information

master code :

7658

SKU :

7658/10

product name :

VU 6028418 hydrochloride

unit size :

10 mg (also 50 mg)

description :

Potent and selective M4 mAChR antagonist

target :

mAChR M4 Antagonists

category :

Small Molecules

purity :

98%

observed molecular weight :

468.95

url print :

?utm_source=labome&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

VU 6028418 hydrochloride is a potent and selective M4 mAChR antagonist (IC50 = 4.1 nM and 57 nM for human and rat M4 respectively). VU 6028418 hydrochloride dose-dependently reduces the latency to withdraw and reverses cataleptic behavior in haloperidol -treated animals. Orally bioavailable.

top caption :

Potent and selective M4 mAChR antagonist

extended description :

Potent and selective M4 mAChR antagonist

chemical name text :

(3aR,5s,6aS)-2-((Tetrahydro-2H-pyran-4-yl)methyl)-N-(6-(2,3,5-trifluorophenyl)pyridazin-3-yl)octahydrocyclopenta[c]pyrrol-5-amine hydrochloride

formula :

C23H27F3N4O.HCl

formula text :

C23H27F3N4O.HCl

USD :

281 USD

product details :

Potent and selective M4 mAChR antagonist

storage :

Store at -20░C

more info or order :

Tocris Bioscience product webpage