7573/10 | Tocris Bioscience 7573/10 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

7573/10

catalog :

7573/10

quantity :

10 mg (also 50 mg)

price :

185 USD

more info or order :

Tocris Bioscience product webpage

image

image 1 :

BAY 1797 CAS No. 2055602-83-8 Selective P2X4 antagonist

product information

master code :

7573

SKU :

7573/10

product name :

BAY 1797

unit size :

10 mg (also 50 mg)

description :

Selective P2X4 antagonist

target :

P2X4

category :

Small Molecules

purity :

98%

observed molecular weight :

416.88

url print :

?utm_source=labome&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

BAY 1797 is a selective purinergic P2X4 receptor antagonist (IC50 values are 108, 112 and 233 nM for the human, mouse and rat P2X4, respectively). It is selective for P2X4 over P2X3, P2X7, and P2X1 receptors (IC50 values are 8.3, 10.6 and 50 M, respectively, for the human receptors). BAY 1797 dose-dependently reduces prostaglandin E2 levels and exhibits anti-inflammatory and analgesic effects in an in vivo model of inflammatory pain. Orally active.

top caption :

Selective P2X4 antagonist

extended description :

Selective P2X4 antagonist

chemical name text :

N-[3-(Aminosulfonyl)-4-(3-chlorophenoxy)phenyl]benzeneacetamide

formula :

C20H17ClN2O4S

formula text :

C20H17ClN2O4S

cas num :

2055602-83-8

USD :

185 USD

product details :

Selective P2X4 antagonist

alt names :

ATP receptor, ATP-gated cation channel protein, P2RX4, P2X purinoceptor 4, P2X4P2X receptor, subunit 4, P2X4R, Purinergic receptor, purinergic receptor P2X, ligand-gated ion channel, 4, purinoceptor P2X4

storage :

Store at -20░C

more info or order :

Tocris Bioscience product webpage