7541/1 | Tocris Bioscience 7541/1 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

7541/1

catalog :

7541/1

quantity :

1 mg

price :

302 USD

more info or order :

Tocris Bioscience product webpage

image

image 1 :

Cat.No. 7541 - Helianorphin-19 Cyclo(Cys-Tyr-Gly-Gly-Phe-Leu-Arg-Arg-Cys-Ile-Arg-Pro-Lys-Leu-Lys) (Disulfide bridge: 1-9)

product information

master code :

7541

SKU :

7541/1

product name :

Helianorphin-19

unit size :

1 mg

description :

Potent and selective G protein-biased opioid receptor (KOR) agonist

target :

Kappa Opioid Receptor Agonists

category :

Peptides

purity :

95%

observed molecular weight :

1790.21

url print :

?utm_source=labome&utm_medium=referral&utm_campaign=product&utm_term=peptides

details of functionality :

Helianorphin-19 is a high affinity, potent and selective G protein-biased -opioid receptor (KOR) agonist (Ki = 25 nM; EC50 = 45 nM). Helianorphin-19 exhibits approximately 200-fold selectivity for KOR over and -opioid receptors. In vivo Helianorphin-19 shows potent peripheral analgesic efficacy in a mouse model of visceral pain without affecting motor coordination/sedation.

top caption :

Potent and selective G protein-biased opioid receptor (KOR) agonist

extended description :

Potent and selective G protein-biased opioid receptor (KOR) agonist

formula :

C81H132N26O16S2

formula text :

C81H132N26O16S2

cas num :

2883653-86-7

USD :

302 USD

product details :

Potent and selective G protein-biased opioid receptor (KOR) agonist

storage :

Store at -20░C

more info or order :

Tocris Bioscience product webpage