7528/5 | Tocris Bioscience 7528/5 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

7528/5

catalog :

7528/5

quantity :

5 mg

price :

330 USD

more info or order :

Tocris Bioscience product webpage

image

image 1 :

Cat.No. 7528 - BSJ-4-116 C40H49ClN8O8S CAS No. 2519823-34-6

product information

master code :

7528

SKU :

7528/5

product name :

BSJ-4-116

unit size :

5 mg

description :

Selective CDK12 PROTAC Degrader

target :

Active Degraders

category :

Small Molecules

purity :

98%

observed molecular weight :

837.39

url print :

?utm_source=labome&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

BSJ-4-116 is a selective CDK12 PROTAC Degrader. BSJ-4-116 selectively degrades CDK12 over a panel of other kinases and exhibits no degradation of CDK13 or cyclin K. The compound inhibits growth of T-ALL cells and sensitizes them to PARP inhibitor Olaparib (Cat. No. 7579). . PROTAC is a registered trademark of Arvinas Operations, Inc., and is used under license.

top caption :

Selective CDK12 PROTAC Degrader

extended description :

Selective CDK12 PROTAC Degrader

chemical name text :

N-[7-[(3R)-3-[[5-Chloro-4-[[2-[(1-methylethyl)sulfonyl]phenyl]amino]-2-pyrimidinyl]amino]-1-piperidinyl]heptyl]-2-[[2-(2,6-dioxo-3-piperidinyl)-2,3-dihydro-1,3-dioxo-1H-isoindol-4-yl]oxy]acetamide

formula :

C40H49ClN8O8S

formula text :

C40H49ClN8O8S

cas num :

2519823-34-6

USD :

330 USD

product details :

Selective CDK12 PROTAC Degrader

storage :

Store at -20░C

more info or order :

Tocris Bioscience product webpage