7493/10 | Tocris Bioscience 7493/10 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

7493/10

catalog :

7493/10

quantity :

10 mg (also 50 mg)

price :

77 USD

more info or order :

Tocris Bioscience product webpage

image

image 1 :

Cat.No. 7493 - Tasimelteon C15H19NO2 CAS No. 609799-22-6

product information

master code :

7493

SKU :

7493/10

product name :

Tasimelteon

unit size :

10 mg (also 50 mg)

description :

Selective dual melatonin receptor (MT1/MT2) agonist

target :

Melatonin (MT) Receptor Agonists

category :

Small Molecules

purity :

98%

observed molecular weight :

245.32

url print :

?utm_source=labome&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Tasimelteon is a high affinity and selective dual melatonin receptor (MT1/MT2) agonist (Ki values are 0.304 nM and 0.0692 nM, respectively). It has no significant interaction with any other commonly screened receptors or enzyme binding sites. Tasimelteon induces a potent, concentration-dependent inhibition of forskolin-stimulated cAMP accumulation in NIH-3T3 cells stably expressing human MT1 (EC50 = 0.74 nM) or expressing human MT2 (EC50 = 0.1 nM) receptors. Tasimelteon is a circadian regulator.

top caption :

Selective dual melatonin receptor (MT1/MT2) agonist

extended description :

Selective dual melatonin receptor (MT1/MT2) agonist

chemical name text :

N-[[(1R,2R)-2-(2,3-Dihydro-4-benzofuranyl)cyclopropyl]methyl]propanamide

formula :

C15H19NO2

formula text :

C15H19NO2

cas num :

609799-22-6

USD :

77 USD

product details :

Selective dual melatonin receptor (MT1/MT2) agonist

storage :

Store at -20░C

more info or order :

Tocris Bioscience product webpage