7159/10 | Tocris Bioscience 7159/10 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

7159/10

catalog :

7159/10

quantity :

10 mg

price :

156 USD

more info or order :

Tocris Bioscience product webpage

image

image 1 :

Cat.No. 7159 - FMF-04-159-R C28H32Cl3N7O5S

product information

master code :

7159

SKU :

7159/10

product name :

FMF-04-159-R

unit size :

10 mg

description :

Potent CDK14 and CDK16 inhibitor; displays reversible inhibition of CDK14

target :

Cyclin-dependent Kinase Inhibitors

category :

Small Molecules

purity :

98%

observed molecular weight :

685.02

url print :

?utm_source=labome&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

FMF-04-159-R is a potent inhibitor of CDK16 and CDK14 (IC50 values are 6 and 140 nM, respectively in kinase activity assay; IC50 = 563 nM for CDK14 in BRET assay). Also binds CDK2 (IC50 = 493 nM). Inhibition reversible upon compound wash-out. Control for FMF-04-159-2 (Cat. No. 7158).

top caption :

Potent CDK14 and CDK16 inhibitor; displays reversible inhibition of CDK14

extended description :

Potent CDK14 and CDK16 inhibitor; displays reversible inhibition of CDK14

chemical name text :

N-(1-((3-(4-(Dimethylamino)butanamido)phenyl)sulfonyl)piperidin-4-yl)-4-(2,4,6-trichlorobenzamido)-1H-pyrazole-3-carboxamide

formula :

C28H32Cl3N7O5S

formula text :

C28H32Cl3N7O5S

cas num :

2741262-15-5

USD :

156 USD

product details :

Potent CDK14 and CDK16 inhibitor; displays reversible inhibition of CDK14

storage :

Store at -20░C

more info or order :

Tocris Bioscience product webpage