7057/10 | Tocris Bioscience 7057/10 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

7057/10

catalog :

7057/10

quantity :

10 mg (also 50 mg)

price :

222 USD

more info or order :

Tocris Bioscience product webpage

image

image 1 :

Cat.No. 7057 - VU 0071063 C18H22N4O2 CAS No. 333415-38-6

product information

master code :

7057

SKU :

7057/10

product name :

VU 0071063

unit size :

10 mg (also 50 mg)

description :

Selective activator of SUR1 Kir6.2 channels

target :

Inward Rectifier Potassium Channel Activators

category :

Small Molecules

purity :

98%

observed molecular weight :

326.4

url print :

?utm_source=labome&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

VU 0071063 is a selective activator of SUR1 Kir6.2 channels and pancreatic -cell KATP channels (EC50 = 7 M and 0.3-10.3 M, respectively). VU 0071063 inhibits insulin secretion in pancreatic -cells by inducing hyperpolarization of -cell membranes and reduces voltage-dependent calcium channel activation and Ca2+ influx. VU 0071063 is active in vivo and brain penetrant.

top caption :

Selective activator of SUR1 Kir6.2 channels

extended description :

Selective activator of SUR1 Kir6.2 channels

chemical name text :

7-[[4-(1,1-Dimethylethyl)phenyl]methyl]-3,7-dihydro-1,3-dimethyl-1H-purine-2,6-dione

formula :

C18H22N4O2

formula text :

C18H22N4O2

cas num :

333415-38-6

USD :

222 USD

product details :

Selective activator of SUR1 Kir6.2 channels

storage :

Store at -20░C

more info or order :

Tocris Bioscience product webpage