A 1899 | Tocris Bioscience 6972/5 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

A 1899

catalog :

6972/5

quantity :

5 mg (also 25 mg)

price :

113 USD

more info or order :

Tocris Bioscience product webpage

image

image 1 :

Cat.No. 6972 - A 1899 C30H26F2N2O3 CAS No. 498577-46-1

product information

brand :

Tocris

master code :

6972

SKU :

6972/5

product name :

A 1899

unit size :

5 mg (also 25 mg)

seo description :

Potent K2P3.1 (TASK-1) and K2P9.1 (TASK-3) blocker

target :

Two-P Potassium Channels Blockers

category :

Small Molecules

purity :

98%

observed molecular weight :

500.55

url print :

?utm_source=biocompare&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

A 1899 is a potent K2P3.1 (TASK-1) and K2P9.1 (TASK-3) channel blocker (IC50 values are 7 nM and 70 nM for human TASK-1 and TASK-3 expressed in CHO cells, respectively). Displays 12.5-fold selectivity for TASK-1 and TASK-3 over other K+ channels (IC50 = 0.9 M for K2P18.1/TRESK and 2 M for all other channels tested). Binds within open channel pore.

top caption :

Potent K2P3.1 (TASK-1) and K2P9.1 (TASK-3) blocker

extended description :

Potent K2P3.1 (TASK-1) and K2P9.1 (TASK-3) blocker

chemical name text :

N-[(2,4-Difluorophenyl)methyl]-2 -[[[2-(4-methoxyphenyl)acetyl]amino]methyl][1,1 -biphenyl]-2-carboxamide

formula :

C30H26F2N2O3

formula text :

C30H26F2N2O3

cas num :

498577-46-1

USD :

113 USD

product details :

Potent K2P3.1 (TASK-1) and K2P9.1 (TASK-3) blocker

storage :

Store at -20░C

more info or order :

Tocris Bioscience product webpage