product summary
Loading...
company name :
Tocris Bioscience
product type :
chemical
product name :
Fenoprofen calcium
catalog :
6926
quantity :
50 mg
price :
90 USD
more info or order :
Tocris Bioscience product webpage
product information
brand :
Tocris
master code :
6926
SKU :
6926/50
product name :
Fenoprofen calcium
description :
Positive allosteric modulator of MC3 receptors; exhibits biased signaling
target :
Melanocortin Receptor Agonists
category :
Small Molecules
unit size :
50 mg
purity :
98%
observed molecular weight :
261.31
url print :
?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules
details of functionality :
Melanocortin 3 (MC3) receptor positive allosteric modulator (PAM; allosteric enhancer) (pEC50 = 8.69); decreases the EC50 of -MSH at MC3R. Stimulates ERK1/2 activation at MC3-5R, with highest ERK1/2 activation observed at 3 and 10 M for MC3R, 1 M for MC4R, and 3 M for MC5R. Exhibits biased signaling at MC3-5R, selectively activating ERK1/2 cascade but not canonical cAMP signaling. Antiarthritic.
catalog number base :
6926
product keywords :
71720-56-4 71720564 Melanocortin 3 MC3 receptor positive allosteric modulators PAMs allosteric enhancers biased signaling antiarthritic anti-inflamatory NSAID Melanocortin Receptors 6926,
extended description :
Positive allosteric modulator of MC3 receptors; exhibits biased signaling
chemical name text :
-Methyl-3-phenoxybenzeneacetic acid hemicalcium salt
formula :
C 15 H 13 O 3 .0.5Ca
formula text :
C15H13O3.0.5Ca
cas num :
34597-40-5
2020 USD :
99
2021 USD :
90 USD
storage :
Store at RT
more info or order :
Tocris Bioscience product webpage
company information
Tocris Bioscience
The Watkins Building
Atlantic Road
Avonmouth, Bristol
BS11 9QD
info@bio-techne.com
https://www.tocris.com
800-343-7475
headquarters: UK