FTBMT | Tocris Bioscience 6784 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

FTBMT

catalog :

6784

quantity :

25 mg

price :

360 USD

more info or order :

Tocris Bioscience product webpage

product information

brand :

Tocris

master code :

6784

SKU :

6784/25

product name :

FTBMT

description :

Potent and selective GPR52 agonist; orally bioavailable and BBB permeable

target :

Orphan 7-TM Receptor Agonists

category :

Small Molecules

unit size :

25 mg

purity :

98%

observed molecular weight :

392.35

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Potent and selective GPR52 agonist (EC50 = 75 nM, Emax = 122%). Selective for GPR52 over a panel of 98 targets including D1, D2, AMPA and NMDA. Suppresses methamphetamine-induced hyperlocomotion in mice. Inhibits MK-801 -induced hyperactivity (model for acute psychosis), without causing catalepsy in mice. Orally bioavailable and brain penetrant.

catalog number base :

6784

product keywords :

GPR52 agonist agonism potent selective Schizophrenia psychosis orally bioavailable and BBB permeable Orphan 7-TM Receptors 6784,

extended description :

Potent and selective GPR52 agonist; orally bioavailable and BBB permeable

chemical name text :

4-[3-[[3-Fluoro-5-(trifluoromethyl)phenyl]methyl]-5-methyl-1H-1,2,4-triazol-1-yl]-2-methylbenzamide

formula :

C 19 H 16 F 4 N 4 O

formula text :

C19H16F4N4O

cas num :

1358575-02-6

2020 USD :

349

2021 USD :

360 USD

storage :

Store at -20°C

more info or order :

Tocris Bioscience product webpage