product summary
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company name :
Tocris Bioscience
product type :
chemical
product name :
FTBMT
catalog :
6784/5
quantity :
5 mg (also 25 mg)
price :
112 USD
more info or order :
image
image 1 :

Cat.No. 6784 - FTBMT C19H16F4N4O CAS No. 1358575-02-6
product information
brand :
Tocris, a Bio-Techne brand
catalog number base :
6784
SKU :
6784/5
product name :
FTBMT
description :
Potent and selective GPR52 agonist; orally bioavailable and BBB permeable
target :
Orphan 7-TM Receptor Agonists
unit size :
5 mg (also 25 mg)
category :
Small Molecules
purity :
98%
storage :
Store at -20°C
observed molecular weight :
392.35
url print :
?utm_source=biocompare&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules
details of functionality :
FTBMT (also known as TP 024) is a potent and selective GPR52 agonist (EC50 = 75 nM, Emax = 122%), which is selective for GPR52 over a panel of 98 targets including D1, D2, AMPA and NMDA. FTBMT suppresses methamphetamine-induced hyperlocomotion in mice, and inhibits MK-801 -induced hyperactivity (model for acute psychosis), without causing catalepsy in mice. This compound is orally bioavailable and brain penetrant.
product keywords :
GPR52 agonist agonism potent selective Schizophrenia psychosis orally bioavailable and BBB permeable TP-024 TP-024 Orphan 7-TM Receptors 6784,
extended description :
Potent and selective GPR52 agonist; orally bioavailable and BBB permeable
chemical name text :
4-[3-[[3-Fluoro-5-(trifluoromethyl)phenyl]methyl]-5-methyl-1H-1,2,4-triazol-1-yl]-2-methylbenzamide
formula :
C19H16F4N4O
formula text :
C19H16F4N4O
cas num :
1358575-02-6
USD :
110
USD 2025 :
112 USD
product details :
Potent and selective GPR52 agonist; orally bioavailable and BBB permeable
alt names :
TP-024
more info or order :
company information

Tocris Bioscience
The Watkins Building
Atlantic Road
Avonmouth, Bristol
BS11 9QD
Atlantic Road
Avonmouth, Bristol
BS11 9QD
info@bio-techne.com
https://www.tocris.com800-343-7475
headquarters: UK
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