ZXH 3-26 | Tocris Bioscience 6713 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

ZXH 3-26

catalog :

6713

quantity :

5 mg

price :

426 USD

more info or order :

Tocris Bioscience product webpage

product information

brand :

Tocris

master code :

6713

SKU :

6713/5

product name :

ZXH 3-26

description :

Potent and selective BRD4 degrader

target :

Active Degraders

category :

Small Molecules

unit size :

5 mg

purity :

98%

observed molecular weight :

785.27

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Potent and selective BRD4 degrader (DC50 5 nM). Exhibits no significant degradation of BRD2 and BRD3. Whole proteome mass spectometry shows significant downregulation of BRD4 only. Active intracellularly.

catalog number base :

6713

product keywords :

ZXH3-26 protacs protac active degraders degrades bromodomains BRD4 potent selective Active Degraders Bromodomains 6713, target protein knockdown, PROTAC, SNIPER

extended description :

Potent and selective BRD4 degrader

chemical name text :

Methyl (6S)-4-(4-chlorophenyl)-2-[[[5-[[2-(2,6-dioxo-3-piperidinyl)-2,3-dihydro-1,3-dioxo-1H-isoindol-4-yl]amino]pentyl]amino]carbonyl]-3,9-dimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetate

formula :

C 38 H 37 ClN 8 O 7 S

formula text :

C38H37ClN8O7S

cas num :

2243076-67-5

2020 USD :

409

2021 USD :

426 USD

storage :

Store at -20°C

more info or order :

Tocris Bioscience product webpage