Ceralifimod | Tocris Bioscience 6690 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

Ceralifimod

catalog :

6690

quantity :

10 mg

price :

123 USD

more info or order :

Tocris Bioscience product webpage

product information

brand :

Tocris

master code :

6690

SKU :

6690/10

product name :

Ceralifimod

description :

Highly potent and selective S1P1 and S1P5 agonist

target :

Sphingosine-1-phosphate Receptor Agonists

category :

Small Molecules

unit size :

10 mg

purity :

95%

observed molecular weight :

435.56

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Highly potent and selective S1P1 and S1P5 agonist (EC50 values are 0.027 and 0.33 nM, respectively, in a cAMP assay). Ki values are 0.574, 0.626, 28.7 5450 and 5630 nM for S1P5, S1P1, S1P4, S1P2, S1P3, respectively. Reduces peripheral lymphocyte count in a mouse EAE model. Orally bioavailable.

catalog number base :

6690

product keywords :

sphingosine-1-phosphate S1P1 S1P5 highly potent selective agonists agonism orally bioavailable Sphingosine-1-phosphate Receptors 6690,

extended description :

Highly potent and selective S1P1 and S1P5 agonist

chemical name text :

1-[[3,4-Dihydro-6-[(2-methoxy-4-propylphenyl)methoxy]-1-methyl-2-naphthalenyl]methyl]-3-azetidinecarboxylic acid

formula :

C 27 H 33 NO 4

formula text :

C27H33NO4

cas num :

891859-12-4

2020 USD :

119

2021 USD :

123 USD

storage :

Store at -20°C

more info or order :

Tocris Bioscience product webpage