GI 530159 | Tocris Bioscience 6689/10 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

GI 530159

catalog :

6689/10

quantity :

10 mg (also 50 mg)

price :

154 USD

more info or order :

Tocris Bioscience product webpage

image

image 1 :

Cat.No. 6689 - GI 530159 C27H20F6N2O2 CAS No. 69563-88-8

product information

brand :

Tocris, a Bio-Techne brand

catalog number base :

6689

SKU :

6689/10

product name :

GI 530159

description :

K2P2.1 (TREK-1) and K2P10.1 (TREK-2) channel activator

target :

Two-P Potassium Channels Activators

unit size :

10 mg (also 50 mg)

category :

Small Molecules

purity :

99%

storage :

Store at +4°C

observed molecular weight :

518.45

url print :

?utm_source=biocompare&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

GI 530159 is a TREK1 and TREK2 channel activator (EC50 = 0.76 M in Rb efflux assay in TREK1-expressing CHO cells). Exhibits selectivity for TREK1/2 over TRAAK, TASK3 and a range of other potassium channels. Hyperpolarizes membrane potential of dorsal root ganglion neurons and depresses neuronal activity in vitro .

product keywords :

GI530159 TREK1 TREK2 channel activators activates K2P2 K2P10 Two-P Potassium Channels 6689,

extended description :

K2P2.1 (TREK-1) and K2P10.1 (TREK-2) channel activator

chemical name text :

4,4 -[[2,2,2-Trifluoro-1-(trifluoromethyl)ethylidene]bis(4,1-phenyleneoxy)]bis[benzenamine]

formula :

C27H20F6N2O2

formula text :

C27H20F6N2O2

cas num :

69563-88-8

USD :

152

USD 2025 :

154 USD

product details :

K2P2.1 (TREK-1) and K2P10.1 (TREK-2) channel activator

more info or order :

Tocris Bioscience product webpage