Tipifarnib | Tocris Bioscience 6410 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

Tipifarnib

catalog :

6410

quantity :

25 mg

price :

405 USD

more info or order :

Tocris Bioscience product webpage

image

image 1 :

Cat.No. 6410 - Tipifarnib C27H22Cl2N4O CAS No. 192185-72-1

product information

brand :

Tocris

master code :

6410

SKU :

6410/25

product name :

Tipifarnib

description :

Potent farnesyltransferase inhibitor; orally bioavailable

target :

Protein Prenyltransferase Inhibitors

category :

Small Molecules

unit size :

25 mg

purity :

98%

observed molecular weight :

489.4

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Potent farnesyltransferase inhibitor. Inhibits farnesylation of lamin B and K-RasB peptide substrates (IC50 values are 0.86 and 7.9 nM, respectively). Inhibits tumor growth in vitro and in vivo . Cell penetrant and orally bioavailable.

catalog number base :

6410

product keywords :

Potent farnesyltransferase inhibitors inhibits antitumor cell penetrant orally bioavailable Protein Prenyltransferases Post-translational Modifications 6410,

extended description :

Potent farnesyltransferase inhibitor; orally bioavailable

chemical name text :

6-[(R)-Amino(4-chlorophenyl)(1-methyl-1H-imidazol-5-yl)methyl}-4-(3-chlorophenyl)-1-methyl-2(1H)-quinolinone

formula :

C 27 H 22 Cl 2 N 4 O

formula text :

C27H22Cl2N4O

cas num :

192185-72-1

2020 USD :

393

2021 USD :

405 USD

storage :

Store at -20°C

more info or order :

Tocris Bioscience product webpage