6372/10 | Tocris Bioscience 6372/10 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

6372/10

catalog :

6372/10

quantity :

10 mg (also 50 mg)

price :

260 USD

more info or order :

Tocris Bioscience product webpage

citations: 1

Reference
Meadows A, Han K, Singh K, Murgia A, McNally B, West J, et al. N-arachidonylglycine is a caloric state-dependent circulating metabolite which regulates human CD4+T cell responsiveness. iScience. 2023;26:106578 pubmed publisher

image

image 1 :

Cat.No. 6372 - PSB CB5 C20H17ClN2O2S CAS No. 1627710-30-8

product information

master code :

6372

SKU :

6372/10

product name :

PSB CB5

unit size :

10 mg (also 50 mg)

description :

Selective GPR18 antagonist

target :

Additional Cannabinoid-related Compounds

category :

Small Molecules

purity :

98%

observed molecular weight :

384.88

url print :

?utm_source=labome&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

PSB CB5 is a selective GPR18 antagonist (IC50 = 0.279 M). Exhibits 36-fold selectivity versus CB1 and GPR55 and 14-fold selectivity versus CB2 receptors. Inhibits N -Arachidonylglycine (Cat. No. 1445) induced acrosomal exocytosis in human spermatozoa.

top caption :

Selective GPR18 antagonist

extended description :

Selective GPR18 antagonist

chemical name text :

(2Z)-2[[3-[(4-Chlorophenyl)methoxy]phenyl]methylene]-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-3(2H)-one

formula :

C20H17ClN2O2S

formula text :

C20H17ClN2O2S

cas num :

1627710-30-8

USD :

260 USD

product details :

Selective GPR18 antagonist

storage :

Store at -20░C

more info or order :

Tocris Bioscience product webpage