TM N1324 | Tocris Bioscience 6325 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

TM N1324

catalog :

6325

quantity :

25 mg

price :

532 USD

more info or order :

Tocris Bioscience product webpage

product information

brand :

Tocris

master code :

6325

SKU :

6325/25

product name :

TM N1324

description :

Potent and selective GPR39 agonist; orally bioavailable

target :

Orphan 7-TM Receptor Agonists

category :

Small Molecules

unit size :

25 mg

purity :

98%

observed molecular weight :

397.79

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Potent and selective GPR39 agonist (IC50 values are 280 and 9 nM in the absence and presence of Zn2+, respectively). Exhibits no significant activity against a panel of 165 other GPCRs. Inhibits the release of ghrelin and somatostatin from primary gastric mucosa cells in vitro . Cell permeable and orally bioavailable.

catalog number base :

6325

product keywords :

TMN1324 gpr39 agonists agonism potent selective orally bioavailable cell permeable zn2+ zinc Orphan 7-TM Receptors 6325,

extended description :

Potent and selective GPR39 agonist; orally bioavailable

chemical name text :

4-(2-Chloro-4-fluorophenyl)-1,4,5,7-tetrahydro-3-methyl-1-(9H-purin-6-yl)-6H-pyrazolo[3,4-b]pyridin-6-one

formula :

C 18 H 13 ClFN 7 O

formula text :

C18H13ClFN7O

cas num :

1144477-35-9

2020 USD :

516

2021 USD :

532 USD

storage :

Store at -20°C

more info or order :

Tocris Bioscience product webpage