6311/10 | Tocris Bioscience 6311/10 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

6311/10

catalog :

6311/10

quantity :

10 mg (also 50 mg)

price :

59 USD

more info or order :

Tocris Bioscience product webpage

image

image 1 :

Cat.No. 6311 - Tadalafil C22H19N3O4 CAS No. 171596-29-5

product information

master code :

6311

SKU :

6311/10

product name :

Tadalafil

unit size :

10 mg (also 50 mg)

description :

Potent and highly selective PDE5 inhibitor; orally bioavailable

target :

Phosphodiesterase Inhibitors

category :

Small Molecules

purity :

99%

observed molecular weight :

389.4

url print :

?utm_source=labome&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Tadalafil is a potent and highly selective PDE5 inhibitor (IC50 = 5 nM). Exhibits 2000-fold selectivity for PDE5 over PDEs 1,2,3 and 4 and 1000-fold selectivity over PDE6. Reduces blood pressure in hypertensive rats. Also delays tumor growth in a mouse model via inhibition of MDSC-mediated immunosuppression. Orally bioavailable.

top caption :

Potent and highly selective PDE5 inhibitor; orally bioavailable

extended description :

Potent and highly selective PDE5 inhibitor; orally bioavailable

chemical name text :

(6R,12aR)-6-(1,3-Benzodioxol-5-yl)-2,3,6,7,12,12a-hexahydro-2-methylpyrazino[1 ,2 :1,6]pyrido[3,4-b]indole-1,4-dione

formula :

C 22 H 19 N 3 O 4

formula text :

C22H19N3O4

cas num :

171596-29-5

USD :

59 USD

product details :

Potent and highly selective PDE5 inhibitor; orally bioavailable

alt names :

GF196960

storage :

Store at -20░C

more info or order :

Tocris Bioscience product webpage