MS 15203 | Tocris Bioscience 6299 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

MS 15203

catalog :

6299

quantity :

25 mg

price :

290 USD

more info or order :

Tocris Bioscience product webpage

product information

brand :

Tocris

master code :

6299

SKU :

6299/25

product name :

MS 15203

description :

Potent and selective GPR171 partial agonist

target :

GPR171 Agonists

category :

Small Molecules

unit size :

25 mg

purity :

98%

observed molecular weight :

249.22

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Potent and selective GPR171 partial agonist (EC50 = 90 nM; 28% inhibition of forskolin activated adenylyl cyclase activity in rat hypothalamic memebranes). Exhibits minimal binding to a panel of ~70 GPCRs and 10 other receptors ( 22% of radioligand displaced from the target receptors). Increases neuronal activity in the paraventricular nucleus. Increases food intake and body weight in mice.

catalog number base :

6299

product keywords :

MS15203 GPR171 agonists agonism food intake body weight GPCR neuropeptide GPR171 6299,

extended description :

Potent and selective GPR171 partial agonist

chemical name text :

5-[(2-Methyl-1-oxo-2-propen-1-yl)amino]-1,3-benzenedicarboxylic acid

formula :

C 12 H 11 NO 5

formula text :

C12H11NO5

cas num :

73912-52-4

2020 USD :

284

2021 USD :

290 USD

storage :

Store at -20°C

more info or order :

Tocris Bioscience product webpage