product summary
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company name :
Tocris Bioscience
product type :
chemical
product name :
L Moses dihydrochloride
catalog :
6251
quantity :
10 mg (also 50 mg)
price :
162 USD
more info or order :
Tocris Bioscience product webpage
product information
brand :
Tocris
master code :
6251
SKU :
6251/10
product name :
L Moses dihydrochloride
description :
High affinity and selective PCAF bromodomain inhibitor
target :
Bromodomain Inhibitors
category :
Small Molecules
unit size :
10 mg (also 50 mg)
purity :
98%
observed molecular weight :
433.38
url print :
?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules
details of functionality :
High affinity and selective cell-permeable p300/CBP-associated factor (PCAF) inhibitor (Ki = 47 nM). Exhibits no significant activity against a panel of 48 other bromodomains except GCN5 (Kd = 600 nM). Exhibits 4500-fold selectivity for PCAF over BRD4. Also exhibits metabolic stability in mouse and human liver microsomes and no observable cytotoxicity in peripheral blood mononuclear cells (PBMC).
catalog number base :
6251
product keywords :
PCAF p300/CBP-associated factor GCN5 general control non-derepressible 5 inhibitors inhibits high affinity selective cell-permeable 2079885-05-3 Bromodomains 6251,
extended description :
High affinity and selective PCAF bromodomain inhibitor
chemical name text :
(1S, 2S)-N1,N1-Dimethyl-N2-(3-methyl-1,2,4-triazolo[3,4-a]phthalazin-6-yl)-1-phenylpropane-1,2-diamine dihydrochloride
formula :
C 21 H 24 N 6 .2HCl
formula text :
C21H24N6.2HCl
2020 USD :
155
2021 USD :
162 USD
storage :
Desiccate at RT
more info or order :
Tocris Bioscience product webpage
company information
Tocris Bioscience
The Watkins Building
Atlantic Road
Avonmouth, Bristol
BS11 9QD
info@bio-techne.com
https://www.tocris.com
800-343-7475
headquarters: UK