EHop 016 | Tocris Bioscience 6248 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

EHop 016

catalog :

6248

quantity :

25 mg

price :

287 USD

more info or order :

Tocris Bioscience product webpage

product information

brand :

Tocris

master code :

6248

SKU :

6248/25

product name :

EHop 016

description :

Rac inhibitor

target :

Rho GTPase Inhibitors

category :

Small Molecules

unit size :

25 mg

purity :

98%

observed molecular weight :

430.55

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Rac inhibitor (IC50 = 1.1 M). Exhibits some selectivity for Rac1 and Rac3 over Cdc42. Blocks the interaction of Rac with guanine nucleotide exchange factor Vav2 in breast cancer cell lines expressing high levels of Rac activity and inhibits activity of Rac downstream effector PAK1. Also inhibits mammary tumor growth and metastasis in mice.

catalog number base :

6248

product keywords :

EHop016 Rac inhibitors inhibits EHop016 Vav2 GEFs guanine nucleotide exchange factors Rac1 Rac3 Rho 6248,

extended description :

Rac inhibitor

chemical name text :

N4-(9-Ethyl-9H-carbazol-3-yl)-N2-[3-(4-morpholinyl)propyl]-2,4-pyrimidinediamine

formula :

C 25 H 30 N 6 O

formula text :

C25H30N6O

cas num :

1380432-32-5

2020 USD :

278

2021 USD :

287 USD

storage :

Store at -20°C

more info or order :

Tocris Bioscience product webpage