SAK 3 | Tocris Bioscience 6239 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

SAK 3

catalog :

6239

quantity :

25 mg

price :

319 USD

more info or order :

Tocris Bioscience product webpage

product information

brand :

Tocris

master code :

6239

SKU :

6239/25

product name :

SAK 3

description :

Potent CaV3.1 and 3.3 activator; orally bioavailable

target :

Voltage-gated Calcium Channel Activators

category :

Small Molecules

unit size :

25 mg

purity :

98%

observed molecular weight :

369.41

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Potent CaV3.1 and CaV3.3 activator. Enhances CaV3.1 and CaV3.3, but not CaV3.2 activity at concentrations of 0.01 - 10 M in neuro2A cells in vitro . Elevates ACh levels in hippocampus. Rescues impaired memory-related behaviors, promotes adult neurogenesis and displays antidepressant-like effects in OBX mice. Orally bioavailable.

catalog number base :

6239

product keywords :

SAK3 voltage-gated Ca2+ channels T-VGCC memory orally bioavailable CaV3.1 Ca3.3 activators activates Cav3.x Channels 6239, Voltage-gated calcium channel activator, voltage gated calcium channel, high-voltage activated Ca2+ channel, high voltage gated ca2+ channel

extended description :

Potent CaV3.1 and 3.3 activator; orally bioavailable

chemical name text :

Ethyl 8 -methyl-2 ,4-dioxo-2-(piperidin-1-yl)-2 H-spiro[cyclopent[2]ene-1,3 -imidazo[1,2-a]pyridine]-3-carboxylate

formula :

C 20 H 23 N 3 O 4

formula text :

C20H23N3O4

cas num :

1256269-87-0

2020 USD :

319

2021 USD :

319 USD

storage :

Store at +4°C

more info or order :

Tocris Bioscience product webpage