6239/5 | Tocris Bioscience 6239/5 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

6239/5

catalog :

6239/5

quantity :

5 mg (also 25 mg)

price :

105 USD

more info or order :

Tocris Bioscience product webpage

product information

master code :

6239

SKU :

6239/5

product name :

SAK 3

unit size :

5 mg (also 25 mg)

description :

Potent CaV3.1 and 3.3 activator; orally bioavailable

target :

Cav3.x Channel Activators

category :

Small Molecules

purity :

98%

observed molecular weight :

369.41

url print :

?utm_source=labome&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

SAK 3 is a potent CaV3.1 and CaV3.3 activator. Enhances CaV3.1 and CaV3.3, but not CaV3.2 activity at concentrations of 0.01 - 10 M in neuro2A cells in vitro . Elevates ACh levels in hippocampus. Rescues impaired memory-related behaviors, promotes adult neurogenesis and displays antidepressant-like effects in OBX mice. Orally bioavailable.

top caption :

Potent CaV3.1 and 3.3 activator; orally bioavailable

extended description :

Potent CaV3.1 and 3.3 activator; orally bioavailable

chemical name text :

Ethyl 8 -methyl-2 ,4-dioxo-2-(piperidin-1-yl)-2 H-spiro[cyclopent[2]ene-1,3 -imidazo[1,2-a]pyridine]-3-carboxylate

formula :

C20H23N3O4

formula text :

C20H23N3O4

cas num :

1256269-87-0

USD :

105 USD

product details :

Potent CaV3.1 and 3.3 activator; orally bioavailable

storage :

Store at +4░C

more info or order :

Tocris Bioscience product webpage