LP 922761 | Tocris Bioscience 6229 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

LP 922761

catalog :

6229

quantity :

10 mg (also 50 mg)

price :

195 USD

more info or order :

Tocris Bioscience product webpage

product information

brand :

Tocris

master code :

6229

SKU :

6229/10

product name :

LP 922761

description :

Potent AAK1 inhibitor; peripherally restricted

target :

Other Kinase Inhibitors

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

98%

observed molecular weight :

410.47

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Potent AAK1 inhibitor (IC50 values are 4.8 and 7.6 nM in enzyme and cell assays, respectively). Exhibits some selectivity for AAK1 over BIKE, and exhibits no significant activity at opioid, adrenergic 2 or GABAA receptors. Orally bioavailable. Peripherally restricted.

catalog number base :

6229

product keywords :

LP922761 AAK1 adapter protein-2 AP2 associated kinase 1 potent inhibitors inhibits peripherally restricted orally bioavailable Other Kinases 6229,

extended description :

Potent AAK1 inhibitor; peripherally restricted

chemical name text :

tert-Butyl (2-((3-(4-carbamoylphenyl)imidazo[1,2-b]pyridazin-6-yl)amino)ethyl)(methyl)carbamate

formula :

C 21 H 26 N 6 O 3

formula text :

C21H26N6O3

cas num :

1454808-95-7

2020 USD :

189

2021 USD :

195 USD

storage :

Store at -20°C

more info or order :

Tocris Bioscience product webpage