J 2156 | Tocris Bioscience 6201/10 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

J 2156

catalog :

6201/10

quantity :

10 mg (also 50 mg)

price :

357 USD

more info or order :

Tocris Bioscience product webpage

image

image 1 :

Cat.No. 6201 - J 2156 C24H28N4O4S.C2HF3O2 CAS No. 2387505-73-7

product information

brand :

Tocris

master code :

6201

SKU :

6201/10

product name :

J 2156

unit size :

10 mg (also 50 mg)

seo description :

Selective high affinity human sst4 agonist

target :

Somatostatin Receptor Agonists

category :

Small Molecules

purity :

98%

observed molecular weight :

582.6

url print :

?utm_source=biocompare&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

J 2156 is a high affinity human somatostatin receptor 4 (sst4) agonist (Ki = 1.2 nM). Displays 400-fold selectivity for human sst4 over other human sst receptor subtypes. Exhibits 2 to 3-fold more potent agonism in vitro than endogenous ligands somatostatin-14 (Cat. No. 1157) and somatostatin-28 (Cat. No. 1165). Reduces inflammatory airway hyperresponsiveness in acute and chronic airway inflammation models in mice. Exhibits anxiolytic effects in elevated plus maze test in mice.

top caption :

Selective high affinity human sst4 agonist

extended description :

Selective high affinity human sst4 agonist

chemical name text :

(1 S,2S)-4-Amino-N-(1 -carbamoyl-2 -phenylethyl)-2-(4 -methyl-1 -naphthalenesulfonylamino)butanamide trifluoroacetate

formula :

C24H28N4O4S.C2HF3O2

formula text :

C24H28N4O4S.C2HF3O2

cas num :

2387505-73-7

USD :

357 USD

product details :

Selective high affinity human sst4 agonist

storage :

Store at -20░C

more info or order :

Tocris Bioscience product webpage