PF 06726304 acetate | Tocris Bioscience 6169 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

PF 06726304 acetate

catalog :

6169

quantity :

10 mg

price :

173 USD

more info or order :

Tocris Bioscience product webpage

product information

brand :

Tocris

master code :

6169

SKU :

6169/10

product name :

PF 06726304 acetate

description :

Highly potent and SAM-competitive EZH2 inhibitor

target :

EZH2 Inhibitor

category :

Small Molecules

unit size :

10 mg

purity :

97%

observed molecular weight :

506.38

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Highly potent and SAM-competitive EZH2 lysine methyltransferase inhibitor (IC50 = 0.7 nM). Inhibits proliferation of Karpas-422 cells (non-Hodgkin s lymphoma) in vitro , and halts tumor growth and reduces intratumoral H3K27Me3 levels in mice.

catalog number base :

6169

product keywords :

PF06726304 acetate highly potent EZH2 inhibitors inhibits enhancer of zeste homolog 2 lysine methyltransferase PRC2 polycomb repressive complex 2 Lysine Methyltransferases EZH2 6169, EZH 2, ENX 1, ENX1, KMT6, KMT 6

extended description :

Highly potent and SAM-competitive EZH2 inhibitor

chemical name text :

5,8-Dichloro-2-[(1,2-dihydro-4,6-dimethyl-2-oxo-3-pyridinyl)methyl]-7-(3,5-dimethyl-4-isoxazolyl)-3,4-dihydro-1(2H)-isoquinolinone acetate

formula :

C 22 H 21 Cl 2 N 3 O 3 .C 2 H 4 O 2

formula text :

C22H21Cl2N3O3.C2H4O2

2020 USD :

173

2021 USD :

173 USD

storage :

Store at RT

more info or order :

Tocris Bioscience product webpage