NVS PAK1 1 | Tocris Bioscience 6132 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

NVS PAK1 1

catalog :

6132

quantity :

25 mg

price :

452 USD

more info or order :

Tocris Bioscience product webpage

product information

brand :

Tocris

master code :

6132

SKU :

6132/25

product name :

NVS PAK1 1

description :

Potent and selective PAK1 inhibitor

target :

PAK Inhibitors

category :

Small Molecules

unit size :

25 mg

purity :

98%

observed molecular weight :

479.93

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Potent and selective PAK1 inhibitor (IC50 = 5 nM). Selective for PAK1 over PAK2 and a panel of 442 kinases. Inhibits autophosphorylation of PAK1 in KRAS-mutated pancreatic cancer cell lines. . Negative control also available.

catalog number base :

6132

product keywords :

NVSPAK11 P21-activated kinases PAK1 inhibitors inhibits potent selective P21-activated Kinases 6132, p21-Activated Kinases, p21-Activated Kinase, PAKs

extended description :

Potent and selective PAK1 inhibitor

chemical name text :

(3S)-3-(2-Chloro-5-(2,2-difluoroethyl)-8-fluoro-5H-dibenzo[b,e][1,4]diazepin-11-ylamino)-N-isopropylpyrrolidine-1-carboxamide

formula :

C 23 H 25 ClF 3 N 5 O

formula text :

C23H25ClF3N5O

cas num :

1783816-74-9

2020 USD :

438

2021 USD :

452 USD

storage :

Store at -20°C

more info or order :

Tocris Bioscience product webpage