product summary
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company name :
Tocris Bioscience
product type :
chemical
product name :
P21d hydrochloride
catalog :
6073
quantity :
5 mg
price :
165 USD
more info or order :
Tocris Bioscience product webpage
product information
brand :
Tocris
master code :
6073
SKU :
6073/5
product name :
P21d hydrochloride
description :
Potent and selective Brk inhibitor
target :
Src Family Kinase Inhibitors
category :
Small Molecules
unit size :
5 mg
purity :
98%
observed molecular weight :
483.93
url print :
?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules
details of functionality :
Potent and selective breast tumor kinase (Brk) inhibitor (IC50 = 30 nM). Exhibits 650-fold selectively for Brk over Aurora B kinase and Lck. Downregulates SNAIL protein, restores E-cadherin expression and suppresses migration in breast cancer cells. Also active in vivo and orally bioavailable.
catalog number base :
6073
product keywords :
Potent selective breast tumor kinase Brk PTK6 inhibitors inhibits orally bioavailable Src Kinases 6073,
extended description :
Potent and selective Brk inhibitor
chemical name text :
[4-[[6-Cyclopropyl-3-(1H-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl]amino]-3-fluorophenyl]-4-morpholinylmethanone hydrochloride
formula :
C 23 H 22 FN 7 O 2 .HCl
formula text :
C23H22FN7O2.HCl
2020 USD :
161
2021 USD :
165 USD
storage :
Store at -20°C
more info or order :
Tocris Bioscience product webpage
company information
Tocris Bioscience
The Watkins Building
Atlantic Road
Avonmouth, Bristol
BS11 9QD
info@bio-techne.com
https://www.tocris.com
800-343-7475
headquarters: UK