TP 472 | Tocris Bioscience 6000/10 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

TP 472

catalog :

6000/10

quantity :

10 mg

price :

249 USD

more info or order :

Tocris Bioscience product webpage

citations: 2

Reference
Yang Q, Bariani M, Falahati A, Khosh A, Lastra R, Siblini H, et al. The Functional Role and Regulatory Mechanism of Bromodomain-Containing Protein 9 in Human Uterine Leiomyosarcoma. Cells. 2022;11: pubmed publisher
Gatchalian J, Malik S, Ho J, Lee D, Kelso T, Shokhirev M, et al. A non-canonical BRD9-containing BAF chromatin remodeling complex regulates naive pluripotency in mouse embryonic stem cells. Nat Commun. 2018;9:5139 pubmed publisher

image

image 1 :

Cat.No. 6000 - TP 472 C20H19N3O2

product information

brand :

Tocris, a Bio-Techne brand

catalog number base :

6000

SKU :

6000/10

product name :

TP 472

description :

Potent BRD9/7 inhibitor

target :

Bromodomain Inhibitors

unit size :

10 mg

category :

Small Molecules

purity :

98%

storage :

Store at -20°C

observed molecular weight :

333.38

url print :

?utm_source=biocompare&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

TP 472 is a potent BRD9/7 inhibitor (Kd values are 33 and 340 nM, respectively) Exhibits 30-fold selectivity for BRD9 over other bromodomains except BRD7. Cell permeable and active in vivo . . Negative Control also available.

product keywords :

TP472 bromodomains BRD9 BRD7 inhibitors potent CAS 2079895-62-6 Bromodomains 6000,

extended description :

Potent BRD9/7 inhibitor

chemical name text :

3-(6-Acetylpyrrolo[1,2-a]pyrimidin-8-yl)-N-cyclopropyl-4-methylbenzamide

formula :

C20H19N3O2

formula text :

C20H19N3O2

cas num :

2079895-62-6

USD :

246

USD 2025 :

249 USD

product details :

Potent BRD9/7 inhibitor

more info or order :

Tocris Bioscience product webpage