PF 04620110 | Tocris Bioscience 5863/5 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

PF 04620110

catalog :

5863/5

quantity :

5 mg (also 25 mg)

price :

107 USD

more info or order :

Tocris Bioscience product webpage

product information

brand :

Tocris

master code :

5863

SKU :

5863/5

rank :

0.0006

product name :

PF 04620110

description :

Potent and selective DGAT-1 inhibitor; orally bioavailable

target :

Diacylglycerol O-Acyltransferase (DGAT) Inhibitors

category :

Small Molecules

sizes available :

5 mg (also 25 mg)

url print :

?utm_source=biocompare&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

PF 04620110 is a potent and selective DGAT-1 inhibitor (IC50 = 19 nM). Exhibits 1000-fold selectivity for DGAT-1 over DGAT-2, and no significant activity against a range of other enzymes, ion channels and receptors. Reduces plasma triglyceride levels in a rat lipid challenge model. Orally bioavailable.

extended description :

Potent and selective DGAT-1 inhibitor; orally bioavailable

chemical name text :

trans-4-[4-(4-Amino-7,8-dihydro-5-oxopyrimido[5,4-f][1,4]oxazepin-6(5H)-yl)phenyl]cyclohexaneacetic acid

formula :

C 21 H 24 N 4 O 4

formula text :

C21H24N4O4

cas num :

1109276-89-2

USD :

107 USD

product details :

Potent and selective DGAT-1 inhibitor; orally bioavailable

storage :

Store the unopened product at 2 - 8 °C. Do not use past expiration date.

more info or order :

Tocris Bioscience product webpage