JZP 361 | Tocris Bioscience 5851/10 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

JZP 361

catalog :

5851/10

quantity :

10 mg (also 50 mg)

price :

135 USD

more info or order :

Tocris Bioscience product webpage

product information

brand :

Tocris

master code :

5851

SKU :

5851/10

rank :

0.0006

product name :

JZP 361

description :

Potent and selective reversible MAGL inhibitor

target :

Monoacylglycerol Lipase Inhibitors

category :

Small Molecules

sizes available :

10 mg (also 50 mg)

url print :

?utm_source=biocompare&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

JZP 361 is a potent and selective reversible MAGL inhibitor (IC50 = 46 nM). Exhibits 35-fold and 150-fold higher selectivity over human FAAH and ABHD6, respectively (IC50 values are 1.79 and 7.24 M, respectively). Displays affinity for H1 receptors (pA2 = 6.81). Exhibits no activity at cannabinoid receptors at 10 M.

extended description :

Potent and selective reversible MAGL inhibitor

chemical name text :

[4-(8-Chloro-5,6-dihydro-11H-benzo[5,6]cyclohepta[1,2-b]pyridin-11-ylidene)-1-piperidinyl](1H-1,2,4-triazol-1-yl)methanone

formula :

C 22 H 20 ClN 5 O

formula text :

C22H20ClN5O

cas num :

1680193-80-9

USD :

135 USD

product details :

Potent and selective reversible MAGL inhibitor

storage :

Store the unopened product at 2 - 8 °C. Do not use past expiration date.

more info or order :

Tocris Bioscience product webpage