LEI 101 hydrochloride | Tocris Bioscience 5826 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

LEI 101 hydrochloride

catalog :

5826

quantity :

10 mg

price :

291 USD

more info or order :

Tocris Bioscience product webpage

product information

brand :

Tocris

master code :

5826

SKU :

5826/10

product name :

LEI 101 hydrochloride

description :

Potent and selective CB2 partial agonist; orally biovailable

target :

Cannabinoid R2/CB2 Agonists

category :

Small Molecules

unit size :

10 mg

purity :

98%

observed molecular weight :

508.99

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Potent and selective CB2 partial agonist (pEC50 = 8.0). Exhibits 100-fold selectivity for CB2 over CB1 and no significant interaction with hFAAH, MAGL, DAGL or NAPE-PLD. Displays antinociceptive activity in a rat neuropathic pain model and attenuates renal inflammation in a mouse kidney damage model. Orally bioavailable with low brain penetration.

catalog number base :

5826

product keywords :

LEI101 hydrochloride cannabinoid CB2 partial agonists potent selective agonism orally bioavailable anti-inflammatory CB2 Receptors 5826,

extended description :

Potent and selective CB2 partial agonist; orally biovailable

chemical name text :

3-Cyclopropyl-1-[[4-[6-[(1,1-dioxido-4-thiomorpholinyl)methyl]-5-fluoro-2-pyridinyl]phenyl]methyl]-2,4-imidazolidinedione hydrochloride

formula :

C 23 H 25 FN 4 O 4 S.HCl

formula text :

C23H25FN4O4S.HCl

cas num :

2250025-91-1

2020 USD :

285

2021 USD :

291 USD

storage :

Store at -20°C

more info or order :

Tocris Bioscience product webpage