GSK 591 dihydrochloride | Tocris Bioscience 5777 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

GSK 591 dihydrochloride

catalog :

5777

quantity :

10 mg

price :

314 USD

more info or order :

Tocris Bioscience product webpage

product information

brand :

Tocris

master code :

5777

SKU :

5777/10

product name :

GSK 591 dihydrochloride

description :

Potent and selective PRMT5 inhibitor

target :

Protein Arginine Methyltransferase Inhibitors

category :

Small Molecules

unit size :

10 mg

purity :

97%

observed molecular weight :

453.41

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Potent and selective PRMT5 inhibitor (IC50 = 4 nM). Selective for PRMT5 over a panel of other PRMTs and lysine methyltransferases. Inhibits proliferation of mantle cell lymphoma (MCL) in vitro . . To request the negative control for GSK 591, please fill out the SGC 2096 request form on the SGC website.

catalog number base :

5777

product keywords :

GSK591 dihydrochloride protein arginine methyltransferases inhibitors inhibits potent selective PRMT5 1616391-87-7 Structural Genomics Consortium SGC GSK3203591 EPZ015866 GSK 3203591 Protein Arginine Methyltransferases 5777,

extended description :

Potent and selective PRMT5 inhibitor

chemical name text :

2-(Cyclobutylamino)-N-[(2S)-3-(3,4-dihydro-2(1H)-isoquinolinyl)-2-hydropropyl]-4-pyridinecarboxamide dihydrochloride

formula :

C 22 H 28 N 4 O 2 .2HCl

formula text :

C22H28N4O2.2HCl

cas num :

2320953-89-5

2020 USD :

304

2021 USD :

314 USD

alt names :

EPZ015866, GSK 3203591

storage :

Desiccate at RT

more info or order :

Tocris Bioscience product webpage