GSK 591 dihydrochloride | Tocris Bioscience 5777/10 product information

This webpage contains legacy information. The product is either no longer available from the supplier or has been delisted at Labome.

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

GSK 591 dihydrochloride

catalog :

5777/10

quantity :

10 mg

price :

375 USD

product information

brand :

Tocris, a Bio-Techne brand

catalog number base :

5777

SKU :

5777/10

product name :

GSK 591 dihydrochloride

description :

Potent and selective PRMT5 inhibitor

target :

Protein Arginine Methyltransferase Inhibitors

unit size :

10 mg

category :

Small Molecules

purity :

97%

storage :

Desiccate at RT

observed molecular weight :

453.41

url print :

?utm_source=biocompare&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

GSK 591 dihydrochloride is a potent and selective PRMT5 inhibitor (IC50 = 4 nM). Selective for PRMT5 over a panel of other PRMTs and lysine methyltransferases. Inhibits proliferation of mantle cell lymphoma (MCL) in vitro . . To request the negative control for GSK 591, please fill out the SGC 2096 request form on the SGC website.

product keywords :

GSK591 dihydrochloride protein arginine methyltransferases inhibitors inhibits potent selective PRMT5 1616391-87-7 Structural Genomics Consortium SGC GSK3203591 EPZ015866 GSK 3203591 Protein Arginine Methyltransferases 5777,

extended description :

Potent and selective PRMT5 inhibitor

chemical name text :

2-(Cyclobutylamino)-N-[(2S)-3-(3,4-dihydro-2(1H)-isoquinolinyl)-2-hydropropyl]-4-pyridinecarboxamide dihydrochloride

formula :

C22H28N4O2.2HCl

formula text :

C22H28N4O2.2HCl

cas num :

2320953-89-5

USD :

371

USD 2025 :

375 USD

product details :

Potent and selective PRMT5 inhibitor

alt names :

EPZ015866,GSK 3203591