AZ 6102 | Tocris Bioscience 5775 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

AZ 6102

catalog :

5775

quantity :

10 mg (also 50 mg)

price :

221 USD

more info or order :

Tocris Bioscience product webpage

product information

brand :

Tocris

master code :

5775

SKU :

5775/10

product name :

AZ 6102

description :

Potent TNKS1/2 inhibitor

target :

Tankyrase Inhibitors

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

98%

observed molecular weight :

428.53

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Potent TNKS2 and TNKS1 inhibitor (IC50 values are 1 and 3 nM, respectively). Exhibits 100-fold selectivity for TNKS1/2 over PARP-1, PARP-2 and PARP-6. Inhibits Wnt signaling in DLD-1 cells (IC50 = 5 nM). Exhibits moderate oral bioavailability.

catalog number base :

5775

product keywords :

AZ6102 potent selective TNKS1 TNKS2 inhibitors inhibits tankyrases Wnt signaling Tankyrase 5775,

extended description :

Potent TNKS1/2 inhibitor

chemical name text :

rel-2-[4-[6-[(3R,5S)-3,5-Dimethyl-1-piperazinyl]-4-methyl-3-pyridinyl]phenyl]-3,7-dihydro-7-methyl-4H-pyrrolo[2,3-d]pyrimidin-4-one

formula :

C 25 H 28 N 6 O

formula text :

C25H28N6O

cas num :

1645286-75-4

2020 USD :

214

2021 USD :

221 USD

storage :

Store at -20°C

more info or order :

Tocris Bioscience product webpage