AZ 6102 | Tocris Bioscience 5775/10 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

AZ 6102

catalog :

5775/10

quantity :

10 mg (also 50 mg)

price :

248 USD

more info or order :

Tocris Bioscience product webpage

image

image 1 :

Cat.No. 5775 - AZ 6102 C25H28N6O CAS No. 1645286-75-4

product information

brand :

Tocris, a Bio-Techne brand

catalog number base :

5775

SKU :

5775/10

product name :

AZ 6102

description :

Potent TNKS1/2 inhibitor

target :

Tankyrase Inhibitors

unit size :

10 mg (also 50 mg)

category :

Small Molecules

purity :

98%

storage :

Store at -20°C

observed molecular weight :

428.53

url print :

?utm_source=biocompare&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

AZ 6102 is a potent TNKS2 and TNKS1 inhibitor (IC50 values are 1 and 3 nM, respectively). Exhibits 100-fold selectivity for TNKS1/2 over PARP-1, PARP-2 and PARP-6. Inhibits Wnt signaling in DLD-1 cells (IC50 = 5 nM). Exhibits moderate oral bioavailability.

product keywords :

AZ6102 potent selective TNKS1 TNKS2 inhibitors inhibits tankyrases Wnt signaling Tankyrase 5775,

extended description :

Potent TNKS1/2 inhibitor

chemical name text :

rel-2-[4-[6-[(3R,5S)-3,5-Dimethyl-1-piperazinyl]-4-methyl-3-pyridinyl]phenyl]-3,7-dihydro-7-methyl-4H-pyrrolo[2,3-d]pyrimidin-4-one

formula :

C25H28N6O

formula text :

C25H28N6O

cas num :

1645286-75-4

USD :

275

USD 2025 :

248 USD

product details :

Potent TNKS1/2 inhibitor

more info or order :

Tocris Bioscience product webpage