AR-C 141990 hydrochloride | Tocris Bioscience 5658 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

AR-C 141990 hydrochloride

catalog :

5658

quantity :

1 mg

price :

253 USD

more info or order :

Tocris Bioscience product webpage

product information

brand :

Tocris

master code :

5658

SKU :

5658/1

product name :

AR-C 141990 hydrochloride

description :

MCT1 inhibitor

target :

Monocarboxylate Transporter Inhibitors

category :

Small Molecules

unit size :

1 mg

purity :

98%

observed molecular weight :

529.05

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Monocarboxylate transporter (MCT1) inhibitor (pKi = 7.6. Exhibits approximately 10-fold selectivity for MCT1 over MCT2 and no significant activity against MCT3 or 4. Inhibits graft versus host response and prolongs cardiac graft survival in a rat model. Immunosuppressant. Also inhibits brain penetration of GHB analog HOCPCA.

catalog number base :

5658

product keywords :

AR-C141990 HCl monocarboxylate transporter 1 MCT1 immunosuppressant graft versus host GvH transplant Monocarboxylate Transporters 5658,

extended description :

MCT1 inhibitor

chemical name text :

5-[[(3R)-3-Hydroxy-1-pyrrolidinyl]carbonyl]-3-methyl-1-(2-methylpropyl)-6-(4-quinolinylmethyl)thieno[2,3-d]pyrimidine-2,4(1H,3H)-dione

formula :

C 26 H 28 N 4 O 4 S.HCl

formula text :

C26H28N4O4S.HCl

2020 USD :

243

2021 USD :

253 USD

storage :

Store at -20°C

more info or order :

Tocris Bioscience product webpage