AZ Dyrk1B 33 | Tocris Bioscience 5632/10 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

AZ Dyrk1B 33

catalog :

5632/10

quantity :

10 mg

price :

332 USD

more info or order :

Tocris Bioscience product webpage

image

image 1 :

Cat.No. 5632 - AZ Dyrk1B 33 C19H16N4 CAS No. 1679330-37-0

product information

brand :

Tocris, a Bio-Techne brand

catalog number base :

5632

SKU :

5632/10

product name :

AZ Dyrk1B 33

description :

Potent and selective Dyrk1B kinase inhibitor

target :

DYRK Inhibitors

unit size :

10 mg

category :

Small Molecules

purity :

98%

storage :

Store at +4°C

observed molecular weight :

300.36

url print :

?utm_source=biocompare&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

AZ Dyrk1B 33 is a potent and selective ATP-competitive Dyrk1B kinase inhibitor (IC50 = 7 nM); displays distinct cellular effects when compared to DYRK1B knockdown through siRNA. Demonstrates cellular in vitro activity (IC50 = 194 nM). Exhibits better selectivity than AZ 191 (Cat. No 5232); displays no off-target effects against a panel of 124 kinases tested (no kinase was inhibited above 50% at 1 M).

product keywords :

AZDyrk1B33 Dyrk1B kinase inhibitors inhibits dual specificity tyrosine phosphorylation regulated kinases potent DYRK 5632,

extended description :

Potent and selective Dyrk1B kinase inhibitor

chemical name text :

3-(2-Methyl-4-pyrimidinyl)-1-(phenylmethyl)-1H-pyrrolo[2,3-c]pyridine

formula :

C19H16N4

formula text :

C19H16N4

cas num :

1679330-37-0

USD :

368

USD 2025 :

332 USD

product details :

Potent and selective Dyrk1B kinase inhibitor

more info or order :

Tocris Bioscience product webpage