product summary
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company name :
Tocris Bioscience
product type :
chemical
product name :
GLPG 0974
catalog :
5621/10
quantity :
10 mg
price :
301 USD
more info or order :
Tocris Bioscience product webpage
product information
brand :
Tocris
master code :
5621
SKU :
5621/10
rank :
0.061
product name :
GLPG 0974
description :
Potent FFA2 (GPR43) antagonist
target :
Free Fatty Acid Receptor Antagonists
category :
Small Molecules
sizes available :
10 mg
url print :
?utm_source=biocompare&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules
details of functionality :
GLPG 0974 is a potent FFA2 antagonist (IC50 = 9 nM). Exhibits selectivity for FFA2 over FFA3. Inhibits acetate-induced human neutrophil migration in plasma or buffer. Also inhibits FFA2-induced expression of CD11b activation-specific epitope (AE) in human whole blood. Orally bioavailable.
extended description :
Potent FFA2 (GPR43) antagonist
chemical name text :
4-[[[(2R)-1-(Benzo[b]thien-3-ylcarbonyl)-2-methyl-2-azetidinyl]carbonyl][(3-chlorophenyl)methyl]amino]butanoic acid
formula :
C 25 H 25 ClN 2 O 4 S
formula text :
C25H25ClN2O4S
cas num :
1391076-61-1
USD :
301 USD
product details :
Potent FFA2 (GPR43) antagonist
storage :
Store the unopened product at 2 - 8 °C. Do not use past expiration date.
more info or order :
Tocris Bioscience product webpage
company information
Tocris Bioscience
The Watkins Building
Atlantic Road
Avonmouth, Bristol
BS11 9QD
info@bio-techne.com
https://www.tocris.com
800-343-7475
headquarters: UK