CINPA 1 | Tocris Bioscience 5605 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

CINPA 1

catalog :

5605

quantity :

10 mg (also 50 mg)

price :

124 USD

more info or order :

Tocris Bioscience product webpage

citations: 1

Reference
Boussadia B, Gangarossa G, Mselli Lakhal L, Rousset M, de Bock F, Lassere F, et al. Lack of CAR impacts neuronal function and cerebrovascular integrity in vivo. Exp Neurol. 2016;283:39-48 pubmed publisher

product information

brand :

Tocris

master code :

5605

SKU :

5605/10

product name :

CINPA 1

description :

Potent CAR antagonist

target :

Constitutive Androstane Receptor Antagonists

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

98%

observed molecular weight :

395.49

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Potent CAR antagonist (IC50 = 70 nM). Exhibits 90-fold selectivity for CAR over pregnane X receptor (PXR). Also selective over a panel of other nuclear receptors including FXR, LXR, PPAR and RXR.

catalog number base :

5605

product keywords :

CINPA1 CAR constitutive androstane receptors potent antagonists Constitutive Androstane Receptor 5605,

extended description :

Potent CAR antagonist

chemical name text :

Ethyl [5-[(diethylamino)acetyl]-10,11-dihydro-5H-dibenz[b,f]azepin-3-yl]carbamate

formula :

C 23 H 29 N 3 O 3

formula text :

C23H29N3O3

cas num :

102636-74-8

2020 USD :

120

2021 USD :

124 USD

storage :

Store at -20°C

more info or order :

Tocris Bioscience product webpage