5584/50 | Tocris Bioscience 5584/50 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

5584/50

catalog :

5584/50

quantity :

50 mg

price :

136 USD

more info or order :

Tocris Bioscience product webpage

citations: 1

Reference
Papon M, Le Feuvre Y, Barreda G xf3 mez G, Favereaux A, Farrugia F, Bouali Benazzouz R, et al. Spinal Inhibition of GABAB Receptors by the Extracellular Matrix Protein Fibulin-2 in Neuropathic Rats. Front Cell Neurosci. 2020;14:214 pubmed publisher

product information

master code :

5584

SKU :

5584/50

product name :

Aripiprazole

unit size :

50 mg

description :

High affinity D2 and 5-HT1A receptor partial agonist; also 5-HT2A antagonist

target :

Dopamine D2 Receptor Agonists

category :

Small Molecules

purity :

99%

observed molecular weight :

448.39

url print :

?utm_source=labome&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Aripiprazole is a high affinity dopamine D2 and 5-HT1A receptor partial agonist (Ki values are ~1.64 and 5.59 nM respectively). Also 5-HT2A antagonist (Ki = 8.7 nM). Suppresses morphine-induced emesis in vivo . Atypical antipsychotic.

top caption :

High affinity D2 and 5-HT1A receptor partial agonist; also 5-HT2A antagonist

extended description :

High affinity D2 and 5-HT1A receptor partial agonist; also 5-HT2A antagonist

chemical name text :

7-[4-[4-(2,3-Dichlorophenyl)-1-piperazinyl]butoxy]-3,4-dihydro-2(1H)-quinolinone

formula :

C23H27Cl2N3O2

formula text :

C23H27Cl2N3O2

cas num :

129722-12-9

USD :

136 USD

product details :

High affinity D2 and 5-HT1A receptor partial agonist; also 5-HT2A antagonist

storage :

Store at -20░C

more info or order :

Tocris Bioscience product webpage