PFI 4 | Tocris Bioscience 5576 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

PFI 4

catalog :

5576

quantity :

10 mg (also 50 mg)

price :

176 USD

more info or order :

Tocris Bioscience product webpage

product information

brand :

Tocris

master code :

5576

SKU :

5576/10

product name :

PFI 4

description :

Potent and selective BRPF1B bromodomain inhibitor

target :

Bromodomain Inhibitors

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

99%

observed molecular weight :

380.44

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Potent and selective BRPF1B bromodomain inhibitor (IC50 = 172 nM). Exhibits 100-fold selectivity for BRPF1 over a panel of other bromodomains including BRPF2 (BRD1), BRPF3 and BRD4. Disrupts BRPF1 binding to histone H3.3. Cell permeable. Inhibits osteoclastogenesis.

catalog number base :

5576

product keywords :

PFI4 potent selective BRPF1 bromodomains epigenetics inhibitors inhibits sgc Bromodomains 5576,

extended description :

Potent and selective BRPF1B bromodomain inhibitor

chemical name text :

N-[2,3-Dihydro-1,3-dimethyl-2-oxo-6-(1-pyrrolidinyl)-1H-benzimidazol-5-yl]-2-methoxybenzamide

formula :

C 21 H 24 N 4 O 3

formula text :

C21H24N4O3

cas num :

900305-37-5

2020 USD :

176

2021 USD :

176 USD

storage :

Store at +4°C

more info or order :

Tocris Bioscience product webpage